Species- or isozyme-specific enzyme inhibitors. 4. Design of a two-site inhibitor of adenylate kinase with isozyme selectivity

J Med Chem. 1982 Jun;25(6):638-44. doi: 10.1021/jm00348a006.
No abstract available

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Adenosine Monophosphate / analogs & derivatives
  • Adenosine Triphosphate / analogs & derivatives
  • Adenylate Kinase / antagonists & inhibitors*
  • Animals
  • Isoenzymes / antagonists & inhibitors*
  • Kinetics
  • Liver / enzymology
  • Muscles / enzymology
  • Phosphotransferases / antagonists & inhibitors*
  • Rabbits
  • Rats
  • Species Specificity
  • Substrate Specificity

Substances

  • Isoenzymes
  • Adenosine Monophosphate
  • Adenosine Triphosphate
  • Phosphotransferases
  • Adenylate Kinase